Basic Peptide Information

DICL ID
DICL_Pep_00196
Ion Channel
Voltage-gated potassium channel subfamily H member 2
Peptide Function
Blocker
Gene Name
KCNH2

Activity Data (nM)

IC50
3.4 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified

Sequence Information

Peptide Sequence
DRDSCVDKSRCAKYGYFQECTDCCKKYGHNGGTCMFFKCKCA
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Not available
Peptide Species
Centruroides margaritatus (Central American bark Scorpion)
Peptide Name
Potassium channel toxin gamma-KTx 1.10
CAS Number
Not available

Experimental Conditions

pH
pH 7.3
Holding Potential (mV)
−120 mV
Temperature
Room Temperture
Test Method
Patch-clamping
Test Species
Not specified

Binding Information

Binding Site
Not specified
Binding Site Residue
Not specified

Ion Channel Information

Gene Abbreviation (ABB)
VGKCs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)

References & Disease Information

Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available